Direct C-H substitution reaction of anilides using hypervalent iodine and their regioselective issues

Kohki Yamamoto; Shinichiro Kamino; Daisuke Sawada

doi:10.1016/j.tetlet.2017.08.079

Direct C-H substitution reaction of anilides using hypervalent iodine and their regioselective issues

Kohki Yamamoto, Shinichiro Kamino, Daisuke Sawada

Research output: Contribution to journal › Article › peer-review

4 Citations (Scopus)

Abstract

The direct C-H substitution reactions of anilides using hypervalent iodine proceeded to afford azide, chloro, bromo, and fluoro derivatives, and their regioselectivity were described. In the specific reaction conditions, the unique regioisomers were obtained.

Original language	English
Pages (from-to)	3936-3938
Number of pages	3
Journal	Tetrahedron Letters
Volume	58
Issue number	41
DOIs	https://doi.org/10.1016/j.tetlet.2017.08.079
Publication status	Published - 2017

Keywords

Anilide substitution
Hypervalent iodine
Regioselective reaction

ASJC Scopus subject areas

Biochemistry
Drug Discovery
Organic Chemistry

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10.1016/j.tetlet.2017.08.079

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title = "Direct C-H substitution reaction of anilides using hypervalent iodine and their regioselective issues",

abstract = "The direct C-H substitution reactions of anilides using hypervalent iodine proceeded to afford azide, chloro, bromo, and fluoro derivatives, and their regioselectivity were described. In the specific reaction conditions, the unique regioisomers were obtained.",

keywords = "Anilide substitution, Hypervalent iodine, Regioselective reaction",

author = "Kohki Yamamoto and Shinichiro Kamino and Daisuke Sawada",

note = "Funding Information: We are grateful for financial support from The Naito Foundation . Publisher Copyright: {\textcopyright} 2017 Elsevier Ltd",

year = "2017",

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language = "English",

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T1 - Direct C-H substitution reaction of anilides using hypervalent iodine and their regioselective issues

AU - Yamamoto, Kohki

AU - Kamino, Shinichiro

AU - Sawada, Daisuke

PY - 2017

Y1 - 2017

N2 - The direct C-H substitution reactions of anilides using hypervalent iodine proceeded to afford azide, chloro, bromo, and fluoro derivatives, and their regioselectivity were described. In the specific reaction conditions, the unique regioisomers were obtained.

AB - The direct C-H substitution reactions of anilides using hypervalent iodine proceeded to afford azide, chloro, bromo, and fluoro derivatives, and their regioselectivity were described. In the specific reaction conditions, the unique regioisomers were obtained.

KW - Anilide substitution

KW - Hypervalent iodine

KW - Regioselective reaction

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M3 - Article

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JO - Tetrahedron Letters

JF - Tetrahedron Letters

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ER -

Direct C-H substitution reaction of anilides using hypervalent iodine and their regioselective issues

Abstract

Keywords

ASJC Scopus subject areas

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